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Darexaban

CAS No. : 365462-23-3

Biological Activity：Darexaban (YM150) is a potent, selective and orally active factor Xa (FXa) inhibitor with an IC₅₀ of 54.6 nM. Darexaban shows high selectivity against other related serine proteases, such as trypsin, thrombin, and kallikrein. Darexaban has anticoagulant and antithrombotic effects^[2]^[3].

Research Area：Cardiovascular Disease

Targets：Factor Xa|Ser/Thr Protease

Related Screening Libraries:Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library Plus;Metabolism/Protease Compound Library;Clinical Compound Library;Drug Repurposing Compound Library;Anti-Cardiovascular Disease Compound Library;Orally Active Compound Library;Human Metabolite Library;Coagulation and Anti-coagulation Compound Library;

Related Small Molecules:SLN124;Chymotrypsin;Bismuth subgallate;SBC-115076;PCSK9-IN-1;APC-6860;Suc-Ile-Glu(γ-pip)-Gly-Arg-pNA hydrochloride;Manusiran;Lanadelumab;PF-06446846 hydrochloride;TP-030-2;Tilpisertib;Bococizumab;Razaxaban hydrochloride;SBC-110736;PCSK9-IN-2;AS(3n-2)-Inclisiran;Recombinant Proteinase K;Pinostrobin;WNK-IN-11-d3;UKI-1;Patamostat;Betrixaban-d6;4-Aminobenzamidine dihydrochloride;Boc-Ile-Glu-Gly-Arg-AMC

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