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Dagrocorat hydrochloride
CAS No. : 1044535-61-6
Biological Activity：Dagrocorat (PF-00251802) hydrochloride is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat hydrochloride is also a time-dependent reversible inhibitor of CYP3A (IC50=1.3 μM in human liver microsomes) and CYP2D6 (Ki=0.57 μM in human liver microsomes). Dagrocorat hydrochloride can be used for the research of rheumatoid arthritis.
Research Area：Endocrinology|Inflammation/Immunology
Targets：Glucocorticoid Receptor|Cytochrome P450
Related Screening Libraries:Bioactive Compound Library Plus;
Related Small Molecules:SR9186;AMG-208;Deflazacort-D5;CYP1B1-IN-1;CYP2C9/CYP2C19-IN-1;Hypericin;Galeterone;Ranitidine;Bergapten;Ginsenoside Rd;AS1810722;Isoglycycoumarin;Glucocorticoid receptor agonist-2;Polygalaxanthone III;Phenyltoloxamine
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