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Astemizole-d3

CAS No. : 1189961-39-4

Biological Activity：Astemizole-d3 is the deuterium labeled Astemizole. Astemizole (R 43512), a second-generation antihistamine drug to diminish allergic symptoms with a long duration of action, is a histamine H1-receptor antagonist, with an IC₅₀ of 4 nM. Astemizole also shows potent hERG K⁺ channel blocking activity with an IC₅₀ of 0.9 nM. Astemizole has antipruritic effects^[2].

Research Area：Inflammation/Immunology|Endocrinology

Targets：Histamine Receptor|Potassium Channel

Related Small Molecules:Kv3 modulator 2;Tripelennamine;Brompheniramine-d6 maleate;Pinacidil;Samelisant;Chlorphenoxamine;AMP-PNP tetralithium;H3 receptor-MO-1;Diphenhydramine;IK1 inhibitor PA-6;ABT-239;VU590;Ketotifen fumarate;Ranitidine;Domiphen bromide;Mesoridazine benzenesulfonate;Tetrandrine;20(S)-Ginsenoside Rg3;Cetirizine;(S)-(+)-Modafinic acid-d5;Diphenylpyraline hydrochloride;Loratadine-d5

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