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SRX246
CAS No. : 512784-93-9
Biological Activity：SRX246 is a potent, CNS-penetrant, highly selective, orally bioavailable vasopressin 1a (V1a) receptor antagonist (Ki=0.3 nM for human V1a). SRX246 has no interaction at V1b and V2 receptors. SRX246 also displays negligible binding at 64 others receptors classes, including 35 G-proteincoupled receptors. SRX246 can be used for treatment of stress-related disorders.
Research Area：Neurological Disease
Targets：Vasopressin Receptor
Related Screening Libraries:Covalent Screening Library Plus;Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Clinical Compound Library;CNS-Penetrant Compound Library;Drug Repurposing Compound Library;Covalent Screening Library;Orally Active Compound Library;Targeted Diversity Library;
Related Small Molecules:Lixivaptan;Mozavaptan hydrochloride;Balovaptan;Big Endothelin-1 (1-38), human;WAY-151932;Felypressin;Antagonist G TFA;Mozavaptan-d6;SKF 100398;Fedovapagon;L-371,257;Argipressin;D[LEU4,LYS8]-VP;d[Cha4]-AVP;RG7713;TASP0390325;Terlipressin-d5;Terlipressin acetate;SR 49059;Big Endothelin-1 (1-39), porcine
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