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GSK137647A

CAS No. : 349085-82-1

Biological Activity：GSK137647A (GSK 137647) is a potent, selective free fatty acid receptor 4 (FFA4) agonist with pEC₅₀ values of 6.3, 6.2, and 6.1 for human, mouse and rat FFA4, and pEC₅₀ values < 4.5 for all three species for FFA1, FFA2, and FFA3, respectively. GSK137647A has anti-inflammatory activity. GSK137647A induces insulin secretion and inhibits epithelial ion transport, GSK137647A is related to regulation of glucose homeostasis and anti-inflammatory response^[2].

Research Area：Metabolic Disease

Targets：Free Fatty Acid Receptor

Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;

Related Small Molecules:GW-1100;Grifolic acid;Ginsenoside Rb2;AP5;GPR40 Activator 1;AM-1638;DC260126;TUG-770;LY2881835;FFA1 agonist-1;GPR120 Agonist 3;AS2034178 free base;GPR40 Agonist 2;BMS-986118;AMG7703;Fasiglifam;MEDICA16;AR420626;AMG 837 sodium salt;Xelaglifam;TUG-1375;GPR120 Agonist 1;GPR40 agonist 5;TUG-424;GPR120 modulator 2;LY2922470;4-CMTB

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