For research use only. We do not sell to patients.
GKA50 quarterhydrate
Biological Activity：GKA50 quarterhydrate is a potent glucokinase activator (EC50=33 nM at 5 mM glucose) and stimulates insulin release from mouse islets of Langerhans. GKA50 quarterhydrate is a glucose-like activator of beta-cell metabolism in rodent and human islets and a Ca2+-dependent modulator of insulin secretion. GKA50 quarterhydrate shows significant glucose lowering in high fat fed female rats[2][3][4].
Research Area：Metabolic Disease
Targets：Glucokinase
Related Small Molecules:PF-04937319;Globalagliatin;Palmitelaidic Acid;Glucokinase activator 1;AZD1656;AMG-3969;RO-28-1675;IHVR-11029;Cadisegliatin;PSN-GK1;Glucokinase activator 3;PF-04991532;Dorzagliatin;AR453588 hydrochloride;AMG-1694;Palmitelaidic acid-d13;BMS-820132;MK-0941 free base;AM-2394
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