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PROTAC AR-V7 degrader-1
CAS No. : 2767440-24-2
Biological Activity：PROTAC AR-V7 degrader-1 (Compound 6) is a potent, orally bioavailable and selective AR-V7 degrader with the DC50 of 0.32 µM by recruiting VHL E3 ligase to Androgen receptor (AR) DNA binding domain (DBD) binder. PROTAC AR-V7 degrader-1 exhibits activity against 22Rv1 cell-line expressing AR-V7 with the EC50 of 0.88 µM.
Research Area：Cancer
Targets：Androgen Receptor|PROTACs
Related Small Molecules:PROTAC Sirt2 Degrader-1;DB0614;VPC-14449;PROTAC VEGFR-2 degrader-2;dTAGV-1-NEG;CCT367766 formic;AC-262536;HDAC6 degrader-1;PROTAC Axl Degrader 2;PhosTAC7;MS98;JPS014;PROTAC PARP1 degrader;MD-224;FKBP12 PROTAC dTAG-7;GTx-007;SJ10542;MS8815;RIP2 Kinase Inhibitor 4;PROTAC EGFR degrader 7;SJ995973;Linuron-d6;CC-885-CH2-PEG1-NH-CH3;MI-136;dFKBP-1;MI-389;BSJ-4-116;MS4078
Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides
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