KZR-504

For research use only. We do not sell to patients.

KZR-504

CAS No. : 1629052-78-3

Biological Activity:KZR-504 is a highly selective inhibitor of immunoproteasome low molecular mass polypeptide 2 (LMP2), with IC50s of 51 nM, 4.274 μM for LMP2 and LMP7, respectively. KZR-504 is of interest for the treatment of autoimmune disease.

Research Area:Inflammation/Immunology

Targets:Proteasome

Related Screening Libraries:Covalent Screening Library Plus;Bioactive Compound Library Plus;Immunology/Inflammation Compound Library;Metabolism/Protease Compound Library;Covalent Screening Library;Ubiquitination Compound Library;Chemical Probe Library;Anti-Blood Cancer Compound Library;

Related Small Molecules:Calpeptin;Calpain Inhibitor VI;MG-101;ONX-0914 TFA;MG-115;UK-101;SAP2-IN-1;LXE408;GSK3494245;PR-39;20S Proteasome-IN-1;M3258;PI-1840;Rpn11-IN-1;Delanzomib;Ac-ANW-AMC;Cyclotheonellazole A;Aclacinomycin A;Vimentin-IN-1;DD1;VR23;Tomatine;Gabexate mesylate;Alicapistat;Neurodegenerative Disorder-Targeting Compound 1

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