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GW9508
CAS No. : 885101-89-3
Biological Activity：GW9508 is a potent and selective G protein-coupled receptors FFA1 (GPR40) and GPR120 agonist with pEC50s of 7.32 and 5.46, respectively. GW9508 shows ~100-fold selectivity for GPR40 over GPR120. GW9508 is inactive against other GPCRs, kinases, proteases, integrins and PPARs. GW9508 is a glucose-sensitive insulin secretagogue and an ATP-sensitive potassium (KATP) channels opener. Anti-inflammatory and anti-atherosclerotic activities[2][3][4].
Research Area：Metabolic Disease|Inflammation/Immunology|Cardiovascular Disease
Targets：Potassium Channel|Free Fatty Acid Receptor
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