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CB1-IN-1
CAS No. : 1429239-98-4
Biological Activity：CB1-IN-1 (BPRCB1184) is a peripherally restricted CB1R antagonist, with Ki of 0.3 nM and 21 nM for CB1R (EC50 = 3 nM) and CB2R, respectively.
IC50 value: 0.3 nM (Ki, CB1R) 21 nM (Ki, CB2R)
Target: CB1R
in vivo: CB1-IN-1 is a novel peripherally restricted cannabinoid 1 receptor antagonist with significant weight-loss efficacy in diet-induced obese mice. CB1-IN-1 has great potential to ameliorate this related metabolic syndrome.
Research Area：Neurological Disease
Targets：Cannabinoid Receptor
Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound Library;Anti-Obesity Compound Library;
Related Small Molecules:Pregnenolone monosulfate sodium;GW842166X;RVD-Hpα TFA;β-Caryophyllene;Hemopressin(rat) TFA;AM8936;Taranabant;Bay 59-3074;NESS 0327;CB1-IN-2;Olivetol;CB1/2 agonist 1;N-Oleoyl glycine;CB1 antagonist 1;COR170;AZD1940;Pregnenolone monosulfate sodium-13C2,d2;MRL-650;Pregnenolone-d4-1;β-Caryophyllene-d2;GAT228;ANEB-001;CBR Agonist-1;BML-190;Tetrahydromagnolol;MJ15;UCM707;2-Arachidonoylglycerol-d8;NIDA-41020
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