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Brexpiprazole hydrochloride
CAS No. : 913612-38-1
Biological Activity：Brexpiprazole (OPC-34712) hydrochloride, an atypical orally active antipsychotic drug, is a partial agonist of human 5-HT1A and dopamine D2L receptor with Kis of 0.12 nM and 0.3 nM, respectively. Brexpiprazole hydrochloride is also a 5-HT2A receptor antagonist with a Ki of 0.47 nM. Brexpiprazole hydrochloride also shows potent antagonist activity at human noradrenergic α1B (Ki=0.17 nM) and α2C receptors (Ki=0.59 nM)[2].
Research Area：Neurological Disease
Targets：Dopamine Receptor|Adrenergic Receptor|5-HT Receptor
Related Small Molecules:F 13714;Alizapride hydrochloride;Thioproperazine;Mosapride-d5;Todralazine;Bromopride-d3;ARC 239 dihydrochloride;Nuciferine;Yohimbine;Glaucine;Salbutamol;Renzapride;SB-277011 dihydrochloride;BI-167107;LY 344864 racemate;Harmine hydrochloride;Talibegron hydrochloride;MIF-1 TFA;Valerenic acid
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