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RTICBM-189

CAS No. : 551909-15-0

Biological Activity：RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB₁) receptor with a pIC₅₀ of 7.54 in Ca²⁺ mobilization assay. RTICBM-189 has pIC₅₀s of 5.29 and 6.25 for hCB₁ and mCB₁, respectively. RTICBM-189 significantly and selectively attenuates the reinstatement of the cocaine-seeking behavior in rats.

Research Area：Neurological Disease

Targets：Cannabinoid Receptor

Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound Library;CNS-Penetrant Compound Library;

Related Small Molecules:Pregnenolone monosulfate sodium;GW842166X;RVD-Hpα TFA;β-Caryophyllene;Hemopressin(rat) TFA;AM8936;Taranabant;Bay 59-3074;NESS 0327;CB1-IN-2;Olivetol;CB1/2 agonist 1;N-Oleoyl glycine;CB1 antagonist 1;COR170;AZD1940;Pregnenolone monosulfate sodium-13C2,d2;MRL-650;Pregnenolone-d4-1;β-Caryophyllene-d2;GAT228;ANEB-001;CBR Agonist-1;BML-190;Tetrahydromagnolol;MJ15;UCM707;2-Arachidonoylglycerol-d8;NIDA-41020

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