2022 - epigenetics modulation frontier

Fulvestrant-9-sulfone-d3

Posted on December 23, 2022 by haoyuan2014

For research use only. We do not sell to patients. Fulvestrant-9-sulfone-d3 Biological Activity：Fulvestrant-9-sulfone-d3 is the deuterium labeled Fulvestrant-9-sulfone. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | […]

Ellipyrone A

Posted on December 23, 2022 by haoyuan2014

For research use only. We do not sell to patients. Ellipyrone A Biological Activity：Ellipyrone A, a γ-pyrone enclosed macrocyclic poyketide, shows inhibition potential against dipeptidyl peptidase-4 (IC50=0.35 mM). Ellipyrone A also has anti-carbolytic property against α-glucosidase (IC50=0.74 mM) and α-amylase (IC50=0.59 mM). Research Area：Metabolic Disease Targets：Dipeptidyl Peptidase Related Small Molecules:Cofrogliptin;Anagliptin-d6;P32/98;Talabostat;Dutogliptin;Gosogliptin;Prodipine hydrochloride;Diprotin B;16-Hydroxycleroda-3,13-dien-15,16-olide;Gemigliptin tartrate;Teneligliptin hydrobromide hydrate;Teneligliptin-d4;DBPR108;Anagliptin hydrochloride;UAMC00039 dihydrochloride;Retagliptin;Diprotin A […]

Afatinib D6

Posted on December 23, 2022 by haoyuan2014

For research use only. We do not sell to patients. Afatinib D6 CAS No. : 1313874-96-2 Biological Activity：Afatinib D6 (BIBW 2992 D6) is deuterium labeled Afatinib. Afatinib (BIBW 2992) is an irreversible EGFR family inhibitor. Research Area：Cancer Targets：EGFR|Autophagy Related Small Molecules:NSC81111;pp60 (v-SRC) Autophosphorylation Site, Phosphorylated;BMS-690514;Osimertinib-13C,d3;EGFR-IN-5;FGFR2-IN-3;Genistein;Epertinib hydrochloride;UNC-CA359;Osimertinib mesylate;AV-412 free base;Nelipepimut-S;Falnidamol;HER2-IN-6;PROTAC EGFR degrader 7;CHMFL-EGFR-202;Avitinib;Naquotinib;Lavendustin A;EAI001;EGFR/HER2/CDK9-IN-2;Cyasterone;DP-C-4;Allitinib Trending products：Recombinant […]

KN-93 hydrochloride

Posted on December 23, 2022 by haoyuan2014

For research use only. We do not sell to patients. KN-93 hydrochloride CAS No. : 1956426-56-4 Biological Activity：KN-93 hydrochloride is a cell-permeable, reversible and competitive inhibitor calmodulin-dependent kinase type II (CaMKII) with a Ki of 370 nM. Research Area：Cancer Targets：Autophagy|CaMK Related Screening Libraries:Bioactive Compound Library Plus;Kinase Inhibitor Library;Neuronal Signaling Compound Library;Anti-Cancer Compound Library;Autophagy Compound Library; […]

(R)-2-((tert-Butoxycarbonyl)amino)pent-4-ynoic acid

Posted on December 23, 2022 by haoyuan2014

For research use only. We do not sell to patients. (R)-2-((tert-Butoxycarbonyl)amino)pent-4-ynoic acid CAS No. : 63039-46-3 Biological Activity：(R)-2-((tert-Butoxycarbonyl)amino)pent-4-ynoic acid is a Glycine (HY-Y0966) derivative. Research Area：Others Targets：Others Related Screening Libraries:Covalent Screening Library Plus; Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries […]

DCEBIO

Posted on December 23, 2022 by haoyuan2014

For research use only. We do not sell to patients. DCEBIO CAS No. : 60563-36-2 Biological Activity：DCEBIO, a derivative of 1-EBIO, is an extremely potent activator of Cl– secretion in T84 colonic cells. DCEBIO stimulates Cl– secretion via the activation of hIK1 K+ channels and the activation of an apical membrane Cl– conductance[2]. Research Area：Inflammation/Immunology […]

EGFR/CSC-IN-1

Posted on December 23, 2022 by haoyuan2014

For research use only. We do not sell to patients. EGFR/CSC-IN-1 Biological Activity：EGFR/CSC-IN-1 is a potential EGFR (IC50 10.52 nM) and cancer stem cell (CSC) dual inhibitor for triple-negative breast cancer treatment. Research Area：Cancer Targets：EGFR Related Small Molecules:NSC81111;pp60 (v-SRC) Autophosphorylation Site, Phosphorylated;BMS-690514;Osimertinib-13C,d3;EGFR-IN-5;FGFR2-IN-3;Genistein;Epertinib hydrochloride;UNC-CA359;Osimertinib mesylate;AV-412 free base;Nelipepimut-S;Falnidamol;HER2-IN-6;PROTAC EGFR degrader 7;CHMFL-EGFR-202;Avitinib;Naquotinib;Lavendustin A;EAI001;EGFR/HER2/CDK9-IN-2;Cyasterone;DP-C-4;Allitinib Trending products：Recombinant Proteins | Bioactive […]

γ-Tocopherol

Posted on December 23, 2022 by haoyuan2014

For research use only. We do not sell to patients. γ-Tocopherol CAS No. : 54-28-4 Biological Activity：γ-Tocopherol (D-γ-Tocopherol) is a potent cyclooxygenase (COX) inhibitor. γ-Tocopherol is a naturally occurring form of Vitamin E in many plant seeds, such as corn oil and soybeans. γ-Tocopherol possesses antiinflammatory properties and anti-cancer activity. Research Area：Cancer|Inflammation/Immunology Targets：Endogenous Metabolite|COX Related […]

DL-Asparagine

Posted on December 23, 2022 by haoyuan2014

For research use only. We do not sell to patients. DL-Asparagine CAS No. : 3130-87-8 Biological Activity：DL-Asparagine is a racemic melange of the Aparagine L and D-enantiomers. DL-Asparagine has been used in growth-media for bacteria-growth. Research Area：Others Targets：Endogenous Metabolite Related Screening Libraries:Natural Product Library Plus;Bioactive Compound Library Plus;Metabolism/Protease Compound Library;Natural Product Library;Human Endogenous Metabolite Compound […]

AE-3763

Posted on December 23, 2022 by haoyuan2014

For research use only. We do not sell to patients. AE-3763 CAS No. : 291778-77-3 Biological Activity：AE-3763 is a peptide-based human neutrophil elastase inhibitor with an IC50 of 29 nM. Research Area：Inflammation/Immunology|Cardiovascular Disease Targets：Elastase Related Screening Libraries:Bioactive Compound Library Plus; Related Small Molecules:Cyclotheonellazole A;JCP174;BAY-678 racemate;Elastase-IN-1;19α-Hydroxyasiatic acid;Tutuilamide A;MDL 101146;Lodelaben;GW311616 hydrochloride;Elastatinal;DMP 777;BAY-85-8501;FK706;SSR69071;Elastase from porcine pancreas;Secologanoside;Tyrosinase/elastase-IN-1;ZD8321;ZD-0892 Trending products：Recombinant […]