Master of Bioactive Molecules | Inhibitors, Screening Libraries & Proteins
For research use only. We do not sell to patients. Felypressin acetate CAS No. : 914453-97-7 Biological Activity：Felypressin acetate (PLV-2 acetate) is a non-catecholamine vasoconstrictor and a vasopressin 1 agonist. Felypressin acetate is widely used in dental procedures[2]. Research Area：Cardiovascular Disease Targets：Vasopressin Receptor Related Screening Libraries:Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library […]
For research use only. We do not sell to patients. PROTAC BRD4 Degrader-2 CAS No. : 2185795-53-1 Biological Activity：PROTAC BRD4 Degrader-2 is a PROTAC connected by ligands for Cereblon and BRD4 with an IC50 of 14.2 nM against BRD4 BD1. Research Area：Cancer Targets：Epigenetic Reader Domain|PROTACs Related Small Molecules:PROTAC Sirt2 Degrader-1;DB0614;RVX-297;BRD4 Inhibitor-19;UNC6349 (Ket2);PROTAC VEGFR-2 degrader-2;Curcumin;GSK6853;dTAGV-1-NEG;CCT367766 formic;GSK4028;SR-0813;HDAC6 […]
For research use only. We do not sell to patients. Thalidomide 4-fluoride CAS No. : 835616-60-9 Biological Activity：Thalidomide 4-fluoride (Cereblon ligand 4) is the Thalidomide-based Cereblon ligand used in the recruitment of CRBN protein. Thalidomide 4-fluoride (Cereblon ligand 4) can be connected to the ligand for IRAK4 protein by a linker to form PROTAC IRAK4 […]
For research use only. We do not sell to patients. Enitociclib CAS No. : 1610358-56-9 Biological Activity：Enitociclib ((+)-Enitociclib) is an enanthiomer of BAY-1251152 with rotation (+). Enitociclib is a potent and selective CDK9 inhibitor with an IC50 of 3 nM. Enitociclib has anti-tumour activity[2]. Research Area：Cancer Targets：CDK Related Screening Libraries:Bioactive Compound Library Plus;Cell Cycle/DNA Damage […]
For research use only. We do not sell to patients. Alamandine CAS No. : 1176306-10-7 Biological Activity：Alamandine, a member of the renin-angiotensin system (RAS), a vasoactive peptide, is an endogenous ligand of the G protein-coupled receptor MrgD. Alamandine targets to protect the kidney and heart through anti-hypertensive actions[2]. Research Area：Cardiovascular Disease Targets：Angiotensin-converting Enzyme (ACE)|Angiotensin Receptor […]
For research use only. We do not sell to patients. alpha-Hederin CAS No. : 27013-91-8 Biological Activity：alpha-Hederin (α-Hederin), a monodesmosidic triterpenoid saponin, exhibits promising antitumor potential against a variety of human cancer cell lines. alpha-Hederin could inhibit the proliferation and induce apoptosis of gastric cancer accompanied by glutathione decrement and reactive oxygen species generation via […]
For research use only. We do not sell to patients. CB2 receptor antagonist 1 CAS No. : 2772693-05-5 Biological Activity：Hexyl resorcinol derivative 29 has been proved to be a CB2 selective competitive antagonist / reverse agonist with good potency. Olivanol and 5- (2-methyloctane-2-yl) resorcinol derivatives 23 and 24 showed significant antinociceptive activity. Compound 24 was […]
For research use only. We do not sell to patients. PKR activator 1 CAS No. : 2283420-62-0 Biological Activity：PKR activator 1 is a potent pyruvate kinase-R (PKR) activator extracted from patent WO2019035865A1, compound E7-93. Research Area：Cardiovascular Disease Targets：Pyruvate Kinase Related Small Molecules:TEPP-46;Etavopivat;Alkannin;PKM2-IN-3;PKM2-IN-1;PKM2 activator 3;PKR-IN-2;PKR activator 2;PKM2 activator 5;Mitapivat;FX-11;PKM2 activator 4;DASA-58;TEPC466;PKM2 activator 2 Trending products：Recombinant Proteins […]
For research use only. We do not sell to patients. (R)-α,α-Diphenylprolinol-d10 hydrochloride Biological Activity：(R)-α,α-Diphenylprolinol-d10 hydrochloride is the deuterium labeled (R)-α,α-Diphenylprolinol hydrochloride. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | […]
For research use only. We do not sell to patients. Allotetrahydrocortisol-d5 CAS No. : 2687961-06-2 Biological Activity：Allotetrahydrocortisol-d5 is the deuterium labeled Allotetrahydrocortisol. Allotetrahydrocortisol (5a-Tetrahydrocortisol) is a metabolite of Cortisol. Cortisol is the main glucocorticoid in human. It is produced in adrenal cortex and plays a crucial role in many physiological processes[2]. Research Area：Others Targets：Endogenous Metabolite […]